منابع مشابه
A facile preparation of trisubstituted amino-furan and -thiophene derivatives.
β-Alkylation of amino-furan and -thiophene heterocycles is described through metal-, acid- and base-free carbon-carbon bond formation. The ability of both heterocycles to undergo selective β-alkylation is compared by mean of experimental and theoretical data. The presence of chiral amine substituents induced the diastereoselective generation of the newly formed additional stereocenter.
متن کاملSynthesis of Furan Derivatives Condensed with Carbohydrates
Eight new furan derivatives have been prepared and characterized. These compounds were obtained by condensation of aminosugar and aminocyclitol intermediates with furan derivatives.
متن کاملFacile synthesis of optically active imidazole derivatives.
Five optically active imidazole derivatives have been synthesized via a facile 4-step reaction sequence starting from commercially available and inexpensive N-Cbz amino acids. While microwave assisted condensation was unsuccessful, the condensation of the corresponding alpha-bromoketones with formamidine acetate in liquid ammonia was revealed to be a useful method for the synthesis of such imid...
متن کاملNano SnCl2-SiO2 Catalyzed Facile Synthesis of Aryloylamido Coumarins Derivatives
A highly efficient and general method for the synthesis of aryloylamido coumarinsderivatives by a three-component condensation of 4-hydroxycoumarin or 4-hydroxy-6-methylpyran-1-one, aryl glyoxals and benzamide in the presence of nano silica supported tin(II) chloride as a heterogeneous catalyst is established. In this method, SnCl2/nano SiO2 wasused as green and reusable catalyst. Excellent yie...
متن کاملThe facile synthesis of a series of tryptophan derivatives
This study reports a facile method for the synthesis of a variety of 5and 6-substituted tryptophan derivatives that are difficult to prepare using alternative enzymatic approaches. Acylation of an activated amino acid, derived from serine in situ, is coupled with an enzymatic resolution step to furnish enantiopure analogues bearing a range of electron withdrawing and releasing substituents. Iso...
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ژورنال
عنوان ژورنال: Chemical and Pharmaceutical Bulletin
سال: 1990
ISSN: 0009-2363,1347-5223
DOI: 10.1248/cpb.38.2581